Best-effort research profile: this record has not passed full two-source scientific verification. Descriptive fields, research protocols, storage/handling notes, and interaction guidance below are shown with their evidence labels, but calculator presets and exact dosing math remain hidden until the record is verified or reaches Community-Supported status.
Quick Facts
Reference Sizes
Not standardized / source review pending
Storage
Use lot-specific analytical and stability documentation
Solubility
Form and salt dependent; verify against the analytical certificate
Best-Effort Research Profile
GW501516 is an investigational PPAR-delta agonist. Early human trials studied lipid endpoints, but development did not produce an approved medicine. Anti-doping authorities warn against its use, and it is prohibited in sport.
Source review pending. This descriptive profile is shown from the available source material as a best-effort educational reference. It has not passed the full verification bar and is not a dosing instruction, medical claim, or treatment recommendation.
Research Profile
Half-Life
No approved-label pharmacokinetic standard
Onset
Trial endpoints were measured over 2 to 12 weeks
Administration Routes (Research)
Oral
Reported Research Effects
PPAR-delta activation
Lipid and metabolic endpoints studied in short human trials
No approved indication
Reported Research Side Effects
No approved therapeutic safety profile
Serious toxicology and development concerns
Prohibited in sport
Data source: Primary literature and authoritative identity records
Reflects preclinical/research literature context only. Not a medical claim, dosing instruction, or treatment recommendation.
Route-Specific Research Protocols
Amounts and schedules are separated by administration route. Evidence badges distinguish labels, human studies, preclinical work, community reports, and evidence gaps.
Label / guidelineHuman studyCommunity onlyPreclinical onlyNot established
OralHuman study only
2.5 mg, 5 mg, or 10 mg daily
Frequency / timing
Once daily
Duration / setting
12 weeks
Technique
Oral
Evidence
Human study protocol
Context: randomized human trial PMID 22814748
Formulation: Oral-mucosal formulations are not dose-equivalent to injectable or topical formulations.
Route safety: Research-study protocol only; it is not an approved or individualized instruction and should not be extrapolated to another route.
Do not convert an amount between routes. Bioavailability, formulation, sterility, monitoring, and clinical context differ by route. Research-use context only; independently verify every cited source.
Research Interactions
Flagged Avoid / Caution Combinations (Research)
Athletic competition
Unsupervised human use
Other investigational metabolic agents
Reflects patterns reported in research/community literature only. Not a safety guarantee, medical advice, or interaction warning for human use.
Research Notes
Cross-reference catalog inclusion confirmed; sales-page dosing was not promoted to a verified protocol without traceable primary evidence.
Supplementary research context only. Not medical advice or a treatment recommendation.
Found a relevant Reddit or forum thread about this compound? Suggest it below. Every suggestion is reviewed by an editor before it appears -- nothing is published automatically.
Related Research Articles
Published articles on this site that mention GW501516 or one of its catalog aliases.
Research Use Only. All content is for educational and research reference only. Not medical advice, a treatment recommendation, or guidance on human use. Compounds are not FDA-approved drugs unless specifically noted.